Biochemistry Questions Biochemistry Questions / Analyse the significance of genetic variations in drug efficacy, using metoprolol's activity changes based on beta-1-adrenergic receptor differences as an example. How can personalized medicine account for these variations in treatment?

Genetic variations between patients can impact the efficacy of a drug. In the case of metoprolol, variations of alleles in the beta-1-adrenergic receptor can result in a very effective response, or no response at all. This is due to alterations in the structure of the receptor, impairing the binding of the drug molecule and thus making it ineffective in some patients.

Clinical genomics can be used to identify patients with specific mutations that make a drug highly effective or ineffective, supporting clinicians in making decisions. This is a form of personalised medicine, allowing quantitative decisions to be made on care pathways.