Analyse the relationship between body fat percentage and drug distribution in the body. |
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Analyse the TGN1412 clinical trial incident and its impact on the safety of biological drug trials. |
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Compare and contrast in vitro testing with in vivo testing in the context of receptor occupancy. |
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Compare and contrast the first generation and second generation antipsychotic drugs. |
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Compare and contrast the mechanisms of action of methotrexate and sulfasalazine as DMARDs for rheumatoid arthritis. |
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Compare and contrast the modulation of GABA_A receptors by benzodiazepines and barbiturates. |
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Compare and contrast the properties of full agonists and partial agonists. |
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Describe the animal models used to study depression and their relevance in assessing the efficacy of antidepressant drugs. |
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Describe the different phases of clinical research in drug development and their respective purposes. |
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Describe the kindling model of epilepsy and how it is used in research. |
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Describe the mechanisms of action of selective serotonin reuptake inhibitors (SSRIs) and the reasons for their slow onset of efficacy. |
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Describe the role of GABA in the treatment of anxiety and the pharmacology of GABA_A receptors. |
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Discuss the challenges of animal toxicology in the development of biopharmaceuticals and propose alternative methods for testing. |
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Discuss the concept of desensitisation and its impact on drug addiction. |
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Discuss the concept of receptor reserve and its impact on agonist binding. |
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Discuss the differences between unipolar depression and bipolar disorder, including their genetic components and brain regions affected. |
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Discuss the different classes of anxiety disorders and the specific treatments for each. |
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Discuss the different types of COX enzymes and their role in the production of inflammatory mediators. |
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Discuss the factors that affect drug absorption through lipid membranes. How does lipid solubility impact pharmacokinetics? |
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Discuss the genetic and environmental factors that contribute to the development of schizophrenia. |
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Discuss the historical significance of opiates as some of the oldest known drugs from plant sources. |
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Discuss the implications of drug competition for plasma protein binding in patients taking multiple medications. |
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Discuss the importance of preclinical development in determining the safety and toxicity of a potential drug. |
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Discuss the importance of receptors as protein targets of drugs and how they can be manipulated by agonists and antagonists. |
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Discuss the physiological effects of benzodiazepine agonists and their therapeutic uses. |
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Discuss the potential side effects of NSAIDs on the gastrointestinal tract and kidneys. |
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Discuss the role of ion channels in the development of epilepsy. |
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Discuss the role of monoamines in depression and how they are targeted by different categories of antidepressant drugs. |
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Discuss the role of the blood-brain barrier in limiting drug distribution to the central nervous system. |
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Evaluate the role of immunotherapies, such as check-point inhibitors and CAR-T therapy, in the treatment of cancer. |
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Examine the concept of immunotoxicology and its implications in drug development. |
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Examine the controversy surrounding the drug VIOXX and its withdrawal from the market. |
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Examine the impact of protein binding on drug concentration and therapeutic effect. |
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Explain how amphetamines and cocaine affect dopamine and noradrenaline levels in the CNS. |
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Explain the concept of pharmacogenomics and its role in personalizing medicine for more effective treatment strategies. |
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Explain the concept of potency and how it is measured in relation to a standard drug. |
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Explain the concept of volume of distribution and how it influences drug distribution in the body. |
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Explain the diagnostic criteria for depression and the role of genetic risk in its development. |
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Explain the difference between a partial seizure and a generalised seizure. |
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Explain the different pathways of dopamine and their functions in the brain. |
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Explain the increasing complexity of biological molecules and provide examples of different forms of biologics. |
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Explain the major side effects associated with monoamine oxidase inhibitors (MAOIs) and the potential risks of combining them with certain foods. |
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Explain the mechanism of action of aspirin as an anti-inflammatory drug and how it differs from other NSAIDs. |
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Explain the mechanism of action of benzodiazepines as antiepileptic drugs. |
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Explain the pharmacokinetics of benzodiazepines and the potential side effects of their use. |
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Explain the process of canonical signalling by GPCRs and how it leads to downstream effector molecule interaction. |
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Explain the process of injecting a virus into the brain to control epilepsy in animal models. |
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Explain the process of target selection in drug discovery and the importance of finding the correct receptor, enzyme, or transport protein. |
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Explain the relationship between drug affinity for receptors and the dose required to obtain 50% occupancy of receptors. |
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Explain the relationship between drug affinity for receptors and the dose required to obtain 50% occupancy of receptors. |
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Explain the role of cytokines and chemokines in the pathogenesis of asthma and how they contribute to the late phase response. |
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Explain the role of enzymes in pharmacology and how inhibitors and prodrugs can affect drug activity. |
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Explain the role of inflammatory mediators in the degradation of joints in rheumatoid arthritis. |
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Explain the significance of post-market surveillance in ensuring drug safety and detecting rare or long-term side effects. |
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Explain the use of animal models in studying anxiety and how behavioural experiments can elicit fear responses. |
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